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New Articles Published in Oct. to Dec. 2015 Cite ChemBridge Screening Compounds and Libraries

San Diego, CA, USA, February 26, 2016/p>

During October through December 2015, more than 30 articles were published that cite the use of ChemBridge small molecule screening compounds or small molecule libraries. The articles cover a wide range of different research areas - a sampling is provided below.

To search the more than 1,400 articles that cite ChemBridge compounds or libraries, visit our Search Page and select to run a Published Compound / Scientific Article search.

  • Repurposing Registered Drugs as Antagonists for Protease-Activated Receptor 2, Journal of Chemical Information and Modeling, PMID 26445028
  • Small Molecule Microarrays Enable the Identification of a Selective, Quadruplex-Binding Inhibitor of MYC Expression, ACS Chemical Biology, PMID 26462961
  • Direct Modulation of Small GTPase Activity and Function, Angewandte Chemie International Edition, PMID 26470842
  • Novel Abscisic Acid Antagonists Identified with Chemical Array Screening, ChemBioChem, PMID 26493545
  • Discovery of 2-Acylaminothiophene-3-Carboxamides as Multitarget Inhibitors for BCR-ABL Kinase and Microtubules, Journal of Chemical Information and Modeling, PMID 26501568
  • Anti-HIV Drug Discovery and Development: Current Innovations and Future Trends, Journal of Medicinal Chemistry, PMID 26509831
  • Identification of a lead like inhibitor of the hepatitis C virus non-structural NS2 autoprotease, Antiviral Research, PMID 26518228
  • Pharmacophore modeling, Virtual Screening, Molecular docking studies and Density Functional theory approaches to identify novel ketohexokinase (KHK) inhibitors, Biosystems, PMID 26521124
  • Omeprazole increases the efficacy of a soluble epoxide hydrolase inhibitor in a PGE2 induced pain model., Toxicology and Applied Pharmacology, PMID 26522832
  • A Chemical Biology Study of Human Pluripotent Stem Cells Unveils HSPA8 as a Key Regulator of Pluripotency, Stem Cell Reports, PMID 26549849
  • Identification of a small-molecule inhibitor of influenza virus via disrupting the subunits interaction of the viral polymerase, Antiviral Research, PMID 26593979
  • Discovery of Small Molecules for Fluorescent Detection of Complement Activation Product C3d, Journal of Medicinal Chemistry, PMID 26613117
  • Exploiting Transient Protein States for the Design of Small-Molecule Stabilizers of Mutant p53, Structure, PMID 26636255
  • Pharmacology and Structural Analysis of Ligand Binding to the Orthosteric Site of Glutamate-Like GluD2 Receptors, Molecular Pharmacology, PMID 26661043
  • Suppression of Drug Resistance in Dengue Virus, mBio, PMID 26670386
  • Selective novel inverse agonists for human GPR43 augment GLP-1 secretion, European Journal of Pharmacology, PMID 26683635
  • UDP-GlcNAc pathway: Potential target for inhibitor discovery against M. tuberculosis, European Journal of Pharmaceutical Sciences, PMID 26690048
  • Nuclear deformability and telomere dynamics are regulated by cell geometric constraints, PNAS, PMID 26699462
  • Mesendogen, anovelinhibitor of TRPM6, promotes mesoderm anddefinitive endoderm differentiationof human embryonicstemcells through alterationof magnesium homeostasis, Heliyon, PMID 26705539
  • Development of CINPA1 analogs as novel and potent inverse agonists of constitutive androstane receptor, European Journal of Medicinal Chemistry, PMID 26717202
  • Identification of B. anthracis N5-carboxyaminoimidazole ribonucleotide mutase (PurE) active site binding compounds via fragment library screening, Bioorganic and Medicinal Chemistry Journal, PMID 26740153
  • Allosteric inhibitors of Coxsackie virus A24 RNA polymerase, Bioorganic and Medicinal Chemistry Journal, PMID 26762834
  • Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666, ACS Medicinal Chemistry Letters
  • Potent and selective N-(4-sulfamoylphenyl)thiourea-based GPR55 agonists, European Journal of Medicinal Chemistry
  • Computer-Aided Drug Discovery Approaches against the Tropical Infectious Diseases Malaria, Tuberculosis, Trypanosomiasis, and Leishmaniasis, ACS Infectious Diseases
  • High-Throughput Screen in Cryptococcus neoformans Identifies a Novel Molecular Scaffold That Inhibits Cell Wall Integrity Pathway Signaling, ACS Infectious Diseases
  • S100B inhibition with duloxetine, a serotonin-norepinephrine reuptake inhibitor, alters macrophage polarization and abrogates glioma growth in mice, Neuro-Oncology
  • Identification of a Potent Inhibitor Targeting Human Lactate Dehydrogenase A and Its Metabolic Modulation for Cancer Cell Line, Bioorganic and Medicinal Chemistry Letters
  • Identification of dual PPARa/c agonists and their effects on lipid metabolism, Bioorganic and Medicinal Chemistry Journal
  • Targeting the Plasmodium vivax equilibrative nucleoside transporter 1 (PvENT1) for antimalarial drug development, International Journal for Parasitology - Drugs and Drug Resistance
  • Potential role of spinal TRPA1 channels in antinociceptive tolerance to 4 spinally administered morphine, Pharmacological Reports

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